List of Kinases for Activity Screening
Table – Kinases for Activity Screening
QuickScout™ Kinase Activity Assays
| Target Name | Group | Available Services | Source (Carna Catalog Number) |
||||||
| (Mobility Shift Assay, IMAP™) | Pre-selected Panel | ||||||||
| ABL (ABL1) | TK | Km bin. | 1 mM | Preincubation | TK | 08-001 | |||
| ABL (ABL1) [E255K] | TK | Km_bin. | 1 mM | Preincubation | 08-094 | ||||
| ABL (ABL1) [T315I] | TK | Km bin. | 1 mM | Preincubation | 08-093 | ||||
| ACK (TNK2) | TK | Km bin. | 1 mM | 08-196 | |||||
| AKT1 | STK | Km bin. | 1 mM | Preincubation | STK | 01-101 | |||
| AKT2 | STK | Km bin. | Preincubation | 01-102 | |||||
| AKT3 | STK | Km bin. | Preincubation | 01-103 | |||||
| ALK | TK | Km bin. | 1 mM | Preincubation | 08-518 | ||||
| ALK [T1151_L1152insT] | TK | Km bin. | 1 mM | 08-539 | |||||
| ALK [C1156Y] | TK | Km bin. | 1 mM | Preincubation | 08-530 | ||||
| ALK [F1174L] | TK | Km bin. | 1 mM | Preincubation | 08-519 | ||||
| ALK [L1196M] | TK | Km bin. | 1 mM | Preincubation | 08-529 | ||||
| ALK [G1202R] | TK | Km bin. | 1 mM | Preincubation | 08-544 | ||||
| ALK [G1269A] | TK | Km bin. | 1 mM | Preincubation | 08-537 | ||||
| ALK [R1275Q] | TK | Km bin. | 1 mM | Preincubation | 08-520 | ||||
| AMPKα1/β1/γ1 (PRKAA1/B1/G1) | STK | Km bin. | 1 mM | Preincubation | STK | 02-113 | |||
| AMPKα2/β1/γ1 (PRKAA2/B1/G1) | STK | Km bin. | Preincubation | 02-114 | |||||
| ARG (ABL2) | TK | Km bin. | 1 mM | Preincubation | 08-102 | ||||
| AurA (AURKA) | STK | Km bin. | 1 mM | Preincubation | STK | Cell_Cycle | 05-101 | ||
| AurA (AURKA)/TPX2 | STK | Km bin. | Preincubation | 05-186 | |||||
| AurB (AURKB)/INCENP | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 05-102 | |||
| AurC (AURKC) | STK | Km bin. | 1 mM | Cell Cycle | 05-103 | ||||
| AXL | TK | Km bin. | 1 mM | 08-107 | |||||
| BLK | TK | Km bin. | 1 mM | 08-164 | |||||
| BMX | TK | Km bin. | 1 mM | Preincubation | 08-179 | ||||
| BRAF | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-122 | |||||
| BRAF [V600E] | STK | 1 mM (Cascade) | 09-144 | ||||||
| BRK (PTK6) | TK | Km bin. | 1 mM | 08-165 | |||||
| BRSK1 | STK | Km bin. | 1 mM | Preincubation | 02-115 | ||||
| BRSK2 | STK | Km bin. | Preincubation | Cell Cycle | 02-116 | ||||
| BTK | TK | Km bin. | 1 mM | 08-180 | |||||
| BTK [C481S] | TK | Km bin. | 1 mM | 08-547 | |||||
| BUB1/BUB3 | STK | Km bin. | Preincubation | 05-187 | |||||
| CaMK1α (CAMK1) | STK | Km bin. | 1 mM | 02-104 | |||||
| CaMK1δ (CAMK1D) | STK | Km bin. | 02-106 | ||||||
| CaMK2α (CAMK2A) | STK | Km bin. | Preincubation | 02-109 | |||||
| CaMK2β (CAMK2B) | STK | Km bin. | Preincubation | 02-110 | |||||
| CaMK2γ (CAMK2G) | STK | Km bin. | Preincubation | 02-112 | |||||
| CaMK2δ (CAMK2D) | STK | Km bin. | Preincubation | 02-111 | |||||
| CaMK4 | STK | Km bin. | 1 mM | Preincubation | STK | 02-108 | |||
| CDC7/ASK | STK | Km bin. | 1 mM | Cell Cycle | 05-109 | ||||
| CDK1 (CDC2)/CycB1 | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 04-102 | |||
| CDK2/CycA2 | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 04-103 | ||
| CDK2/CycE1 | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 04-165 | |||
| CDK3/CycE1 | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 04-104 | |||
| CDK4/CycD3 | STK | Km bin. | 1 mM | Cell Cycle | 04-105 | ||||
| CDK5/p25 | STK | Km bin. | 1 mM | Preincubation | 04-106 | ||||
| CDK6/CycD3 | STK | Km bin. | 1 mM | Cell Cycle | 04-107 | ||||
| CDK7/CycH/MAT1 | STK | Km bin. | 1 mM | Cell Cycle | 04-108 | ||||
| CDK9/CycT1 | STK | Km bin. | 1 mM | Cell Cycle | 04-110 | ||||
| CGK2 (PRKG2) | STK | Km bin. | Preincubation | 01-143 | |||||
| CHK1 (CHEK1) | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 02-117 | ||
| CHK2 (CHEK2) | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 02-162 | |||
| CK1α (CSNK1A1) | STK | Km bin. | 1 mM | 03-101 | |||||
| CK1γ2 (CSNK1G1) | STK | Km bin. | Preincubation | 03-105 | |||||
| CK1γ2 (CSNK1G2) | STK | Km bin. | Preincubation | 03-106 | |||||
| CK1γ3 (CSNK1G3) | STK | Km bin. | Preincubation | 03-107 | |||||
| CK1δ (CSNK1D) | STK | Km bin. | Preincubation | 03-103 | |||||
| CK1ε (CSNK1E) | STK | Km bin. | 1 mM | STK | 03-104 | ||||
| CK2α1/β (CSNK2A1/B) | STK | Km bin. | 1 mM | Preincubation | Cell Cycle | 05-184 | |||
| CK2α2/β (CSNK2A2/B) | STK | Km bin. | Preincubation | Cell Cycle | 05-185 | ||||
| CLK1 | STK | Km bin. | 1 mM | Preincubation | 04-126 | ||||
| CLK2 | STK | Km bin. | 1 mM | Preincubation | 04-127 | ||||
| CLK3 | STK | Km bin. | Preincubation | 04-128 | |||||
| COT (MAP3K8) | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-301 | |||||
| CRIK (CIT) | STK | Km bin. | 01-104 | ||||||
| CSK | TK | Km bin. | 1 mM | TK | 08-111 | ||||
| DAPK1 | STK | Km bin. | 1 mM | Preincubation | STK | 02-134 | |||
| DCAMKL2 | STK | Km bin. | 02-140 | ||||||
| DDR1 | TK | Km bin. | 1 mM | 08-113 | |||||
| DDR2 | TK | Km bin. | 1 mM | 08-114 | |||||
| DLK (MAP3K12) | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-111 | |||||
| DYRK1A | STK | Km bin. | 1 mM | Preincubation | 04-130 | ||||
| DYRK1B | STK | Km bin. | 1 mM | Preincubation | STK | 04-131 | |||
| DYRK2 | STK | Km bin. | Preincubation | 04-132 | |||||
| DYRK3 | STK | Km bin. | Preincubation | 04-133 | |||||
| EEF2K | STK | Km bin. | 10-113 | ||||||
| EGFR | TK | Km bin. | 1 mM | Preincubation | TK | 08-115 | |||
| EGFR [d746-750] | TK | Km bin. | 1 mM | Preincubation | 08-527 | ||||
| EGFR [d746-750/T790M] | TK | Km bin. | 1 mM | 08-528 | |||||
| EGFR [d746-750/T790M/C797S] | TK | Km bin. | 1 mM | 08-565 | |||||
| EGFR [d746-750/C797S] | TK | Km bin. | 1 mM | Preincubation | 08-564 | ||||
| EGFR[D770_N771insNPG] | TK | Km bin. | 1 mM | 08-553 | |||||
| EGFR [T790M] | TK | Km bin. | 1 mM | Preincubation | 08-194 | ||||
| EGFR [T790M/L858R] | TK | Km bin. | 1 mM | Preincubation | 08-510 | ||||
| EGFR [T790M/C797S/L858R] | TK | 1 mM | 08-510 | ||||||
| EGFR [C797S/L858R] | TK | Km bin. | 1 mM | 08-510 | |||||
| EGFR [L858R] | TK | Km bin. | 1 mM | Preincubation | 08-502 | ||||
| EGFR [L861Q] | TK | Km bin. | 1 mM | Preincubation | 08-513 | ||||
| EML4-ALK | TK | Km bin. | 1 mM | 08-516 | |||||
| EPHA1 | TK | Km bin. | 1 mM | Preincubation | 08-119 | ||||
| EPHA2 | TK | Km bin. | 1 mM | Preincubation | TK | 08-121 | |||
| EPHA3 | TK | Km bin. | 1 mM | Preincubation | 08-122 | ||||
| EPHA4 | TK | Km bin. | 1 mM | Preincubation | 08-123 | ||||
| EPHA5 | TK | Km bin. | 1 mM | Preincubation | 08-124 | ||||
| EPHA6 | TK | Km bin. | 1 mM | Preincubation | 08-125 | ||||
| EPHA7 | TK | Km bin. | 1 mM | Preincubation | 08-126 | ||||
| EPHA8 | TK | Km bin. | 1 mM | Preincubation | 08-127 | ||||
| EPHB1 | TK | Km bin. | 1 mM | Preincubation | 08-128 | ||||
| EPHB2 | TK | Km bin. | 1 mM | Preincubation | 08-129 | ||||
| EPHB3 | TK | Km bin. | 1 mM | Preincubation | 08-130 | ||||
| EPHB4 | TK | Km bin. | 1 mM | Preincubation | TK | 08-131 | |||
| Erk1 (MAPK3) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-142 | |||
| Erk2 (MAPK1) | STK | Km bin. | 1 mM | Preincubation | STK | MAPK (Cascade) | 04-143 | ||
| Erk5 (MAPK7) | STK | Km bin. | 1 mM | MAPK (Cascade) | 04-146 | ||||
| FAK (PTK2) | TK | Km bin. | 1 mM | 08-137 | |||||
| FER | TK | Km bin. | 1 mM | Preincubation | 08-139 | ||||
| FES | TK | Km bin. | 1 mM | Preincubation | 08-140 | ||||
| FGFR1 | TK | Km bin. | 1 mM | Preincubation | TK | 08-133 | |||
| FGFR1 [V561M] | TK | Km bin. | 1 mM | 08-536 | |||||
| FGFR2 | TK | Km bin. | 1 mM | Preincubation | 08-134 | ||||
| FGFR2 [V564I] | TK | Km bin. | 1 mM | Preincubation | 08-546 | ||||
| FGFR3 | TK | Km bin. | 1 mM | 08-135 | |||||
| FGFR3 [V555L] | TK | Km bin. | 1 mM | 08-548 | |||||
| FGFR3 [K650E] | TK | Km bin. | 1 mM | 08-501 | |||||
| FGFR3 [K650M] | TK | Km bin. | 1 mM | 08-199 | |||||
| FGFR3 [V555M] | TK | Km bin. | 1 mM | 08-543 | |||||
| FGFR4 | TK | Km bin. | 1 mM | Preincubation | 08-136 | ||||
| FGFR4 [N535K] | TK | Km bin. | 1 mM | 08-524 | |||||
| FGFR4 [V550E] | TK | Km bin. | 1 mM | 08-525 | |||||
| FGFR4 [V550L] | TK | Km bin. | 1 mM | Preincubation | 08-526 | ||||
| FGR | TK | Km bin. | 1 mM | Preincubation | 08-166 | ||||
| FLT1 | TK | Km bin. | 1 mM | Preincubation | 08-189 | ||||
| FLT3 | TK | Km bin. | 1 mM | TK | 08-154 | ||||
| FLT4 | TK | Km bin. | 1 mM | Preincubation | 08-190 | ||||
| FMS (CSF1R) | TK | Km bin. | 1 mM | 08-155 | |||||
| FRK | TK | Km bin. | 1 mM | Preincubation | 08-167 | ||||
| FYN [isoform a] | TK | Km bin. | 1 mM | 08-168 | |||||
| FYN [isoform b] | TK | Km bin. | 1 mM | 08-531 | |||||
| GSK3α (GSK3A) | STK | Km bin. | 1 mM | Preincubation | 04-140 | ||||
| GSK3β (GSK3B) | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 04-141 | ||
| Haspin (GSG2) | STK | Km bin. | Preincubation | 05-111 | |||||
| HCK | TK | Km bin. | 1 mM | 08-169 | |||||
| HER2 (ERBB2) | TK | Km bin. | 1 mM | 08-016 | |||||
| HER4 (ERBB4) | TK | Km bin. | 1 mM | Preincubation | 08-118 | ||||
| HGK (MAP4K4) | STK | Km bin. | 1 mM | STK | 07-137 | ||||
| HIPK1 | STK | Km bin. | Preincubation | 04-135 | |||||
| HIPK2 | STK | Km bin. | Preincubation | 04-136 | |||||
| HIPK3 | STK | Km bin. | Preincubation | 04-137 | |||||
| HIPK4 | STK | Km bin. | 1 mM | Preincubation | 04-138 | ||||
| HPK1 (MAP4K1) | STK | Km bin. | 07-410 | ||||||
| IGF1R | TK | Km bin. | 1 mM | Preincubation | TK | 08-141 | |||
| IKKα (CHUK) | STK | Km bin. | 05-112 | ||||||
| IKKβ (IKBKB) | STK | Km bin. | 1 mM | Preincubation | STK | 05-084 | |||
| IKKε (IKBKE) | STK | Km bin. | 05-114 | ||||||
| INSR | TK | Km bin. | 1 mM | Preincubation | 08-142 | ||||
| IRAK1 | STK | Km bin. | 09-101 | ||||||
| IRAK4 | STK | Km bin. | 1 mM | STK | 09-145 | ||||
| IRR (INSRR) | TK | Km bin. | 1 mM | 08-143 | |||||
| ITK | TK | Km bin. | 1 mM | TK | 08-181 | ||||
| JAK1 | TK | Km bin. | 1 mM | 08-144 | |||||
| JAK2 | TK | Km bin. | 1 mM | Preincubation | 08-045 | ||||
| JAK3 | TK | Km bin. | 1 mM | Preincubation | TK | 08-046 | |||
| JNK1 (MAPK8) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-163 | |||
| JNK2 (MAPK9) | STK | Km bin. | 1 mM | Preincubation | STK | MAPK (Cascade) | 04-164 | ||
| JNK3 (MAPK10) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-150 | |||
| KDR (VEGFR2) | TK | Km bin. | 1 mM | Preincubation | TK | 08-191 | |||
| KIT | TK | Km bin. | 1 mM | 08-156 | |||||
| KIT [V560G] | TK | Km bin. | 1 mM | 08-504 | |||||
| KIT [V654A] | TK | Km bin. | 1 mM | 08-511 | |||||
| KIT [T670I] | TK | Km bin. | 1 mM | 08-195 | |||||
| KIT [D816E] | TK | Km bin. | 1 mM | 08-541 | |||||
| KIT [D816V] | TK | Km bin. | 1 mM | 08-505 | |||||
| KIT [D816Y] | TK | Km bin. | 1 mM | 08-534 | |||||
| LATS1/MOBKL1A | STK | Km bin. | 01-523 | ||||||
| LATS2/MOBKL1A | STK | Km bin. | 01-524 | ||||||
| LCK | TK | Km bin. | 1 mM | Preincubation | TK | 08-170 | |||
| LOK (STK10) | STK | Km bin. | 07-315 | ||||||
| LTK | TK | Km bin. | 1 mM | 08-106 | |||||
| LYNa | TK | Km bin. | 1 mM | Preincubation | 08-171 | ||||
| LYNb | TK | Km bin. | 1 mM | Preincubation | 08-172 | ||||
| MAP2K1 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-141 | |||||
| MAP2K2 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-142 | |||||
| MAP2K3 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-143 | |||||
| MAP2K4 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-144 | |||||
| MAP2K5 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-145 | |||||
| MAP2K6 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-146 | |||||
| MAP2K7 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-148 | |||||
| MAP3K1 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-103 | |||||
| MAP3K2 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-104 | |||||
| MAP3K3 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-105 | |||||
| MAP3K4 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-106 | |||||
| MAP3K5 | STK | 1 mM (Cascade) | MAPK (Cascade) | 07-107 | |||||
| MAP4K2 | STK | Km bin. | 07-111 | ||||||
| MAPKAPK2 | STK | Km bin. | 1 mM | Preincubation | STK | 02-142 | |||
| MAPKAPK3 | STK | Km bin. | Preincubation | 02-143 | |||||
| MAPKAPK5 | STK | Km bin. | Preincubation | 02-144 | |||||
| MARK1 | STK | Km bin. | Preincubation | 02-120 | |||||
| MARK2 | STK | Km bin. | Preincubation | 02-121 | |||||
| MARK3 | STK | Km bin. | Preincubation | 02-122 | |||||
| MARK4 | STK | Km bin. | Preincubation | 02-123 | |||||
| MELK | STK | Km bin. | 02-124 | ||||||
| MER (MERTK) | TK | Km bin. | 1 mM | Preincubation | 08-108 | ||||
| MET | TK | Km bin. | 1 mM | Preincubation | TK | 08-151 | |||
| MET [D1228H] | TK | Km bin. | 1 mM | Preincubation | 08-540 | ||||
| MET [Y1235D] | TK | Km bin. | 1 mM | Preincubation | 08-198 | ||||
| MET [M1250T] | TK | Km bin. | 1 mM | Preincubation | 08-545 | ||||
| MINK (MINK1) | STK | Km bin. | 1 mM | 07-139 | |||||
| MLK1 (MAP3K9) | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-115 | |||||
| MLK2 (MAP3K10) | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-116 | |||||
| MLK3 (MAP3K11) | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-017 | |||||
| MNK1 (MKNK1) | STK | Km bin. | Preincubation | 02-145 | |||||
| MNK2 (MKNK2) | STK | Km bin. | Preincubation | 02-146 | |||||
| MOS | STK | 1 mM (Cascade) | MAPK (Cascade) | 05-118 | |||||
| MRCKα (CDC42BPA) | STK | Km bin. | 01-107 | ||||||
| MRCKβ (CDC42BPB) | STK | Km bin. | 01-108 | ||||||
| MSK1 (RPS6KA5) | STK | Km bin. | Preincubation | 01-147 | |||||
| MSK2 (RPS6KA4) | STK | Km bin. | 01-148 | ||||||
| MSSK1 (STK23) | STK | Km bin. | 04-159 | ||||||
| MST1 (STK4) | STK | Km bin. | 1 mM | STK | 07-116 | ||||
| MST2 (STK3) | STK | Km bin. | 07-117 | ||||||
| MST3 (STK24) | STK | Km bin. | 07-118 | ||||||
| MST4 | STK | Km bin. | 07-119 | ||||||
| MUSK | TK | Km bin. | 1 mM | 08-153 | |||||
| NDR1 (STK38) | STK | Km bin. | 01-125 | ||||||
| NDR2 (STK38L) | STK | Km bin. | 01-126 | ||||||
| NEK1 | STK | Km bin. | 1 mM | Cell Cycle | 05-123 | ||||
| NEK2 | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 05-226 | ||
| NEK4 | STK | Km bin. | Preincubation | 05-128 | |||||
| NEK6 | STK | Km bin. | 1 mM | Cell Cycle | 05-130 | ||||
| NEK7 | STK | Km bin. | 1 mM | Cell Cycle | 05-131 | ||||
| NEK9 | STK | Km bin. | 1 mM | Cell Cycle | 05-133 | ||||
| NIM1K (MGC42105) | STK | Km bin. | Preincubation | 02-175 | |||||
| NPM1-ALK | TK | Km bin. | 1 mM | Preincubation | 08-517 | ||||
| NuaK1 (ARK5) | STK | Km bin. | Preincubation | 02-126 | |||||
| NuaK2 | STK | Km bin. | Preincubation | 02-127 | |||||
| p38α (MAPK14) | STK | Km bin. | 1 mM | Preincubation | STK | MAPK (Cascade) | Cell Cycle | 04-152 | |
| p38β (MAPK11) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-153 | |||
| p38γ (MAPK12) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-155 | |||
| p38δ (MAPK13) | STK | Km bin. | 1 mM | Preincubation | MAPK (Cascade) | 04-154 | |||
| p70S6K (RPS6KB1) | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 01-154 | ||
| p70S6Kβ (RPS6KB2) | STK | Km bin. | Preincubation | 01-155 | |||||
| PAK1 | STK | Km bin. | Preincubation | 07-123 | |||||
| PAK2 | STK | Km bin. | 1 mM | Preincubation | STK | 07-124 | |||
| PAK4 | STK | Km bin. | 07-126 | ||||||
| PAK5 (PAK7) | STK | Km bin. | Preincubation | 07-127 | |||||
| PAK6 | STK | Km bin. | 07-128 | ||||||
| PASK | STK | Km bin. | 02-128 | ||||||
| PBK | STK | Km bin. | 1 mM | STK | 05-168 | ||||
| PDGFRα (PDGFRA) | TK | Km bin. | 1 mM | Preincubation | TK | 08-157 | |||
| PDGFRα (PDGFRA) [V561D] | TK | Km bin. | 1 mM | Preincubation | 08-507 | ||||
| PDGFRα (PDGFRA) [T674I] | TK | Km bin. | 1 mM | 08-503 | |||||
| PDGFRα (PDGFRA) [D842V] | TK | Km bin. | 1 mM | Preincubation | 08-506 | ||||
| PDGFRβ (PDGFRB) | TK | Km bin. | 1 mM | Preincubation | 08-158 | ||||
| PDHK2 (PDK2) | STK | Km bin. | 10-140 | ||||||
| PDHK4 (PDK4) | STK | Km bin. | 10-125 | ||||||
| PDK1 (PDPK1) | STK | Km bin. | 1 mM | STK | 01-132 | ||||
| PEK (EIF2AK3) | STK | Km bin. | 05-155 | ||||||
| PGK (PRKG1) | STK | Km bin. | 01-142 | ||||||
| PHKG1 | STK | Km bin. | 02-152 | ||||||
| PHKG2 | STK | Km bin. | 02-153 | ||||||
| PIM1 | STK | Km bin. | 1 mM | Preincubation | STK | Cell Cycle | 02-054 | ||
| PIM2 | STK | Km bin. | 1 mM | Cell Cycle | 02-155 | ||||
| PIM3 | STK | Km bin. | 02-156 | ||||||
| PKACα (PRKACA) | STK | Km bin. | 1 mM | STK | 01-127 | ||||
| PKACβ (PRKACB) | STK | Km bin. | 01-128 | ||||||
| PKACγ (PRKACG) | STK | Km bin. | 01-129 | ||||||
| PKCα (PRKCA) | STK | Km bin. | 1 mM | STK | 01-133 | ||||
| PKCβ1 (PRKCB1) | STK | Km bin. | 01-134 | ||||||
| PKCβ2 (PRKCB2) | STK | Km bin. | 01-165 | ||||||
| PKCγ (PRKCG) | STK | Km bin. | 01-137 | ||||||
| PKCδ (PRKCD) | STK | Km bin. | Preincubation | 01-135 | |||||
| PKCε (PRKCE) | STK | Km bin. | 1 mM | Preincubation | 01-136 | ||||
| PKCζ (PRKCZ) | STK | Km bin. | Preincubation | 01-141 | |||||
| PKCη (PRKCH) | STK | Km bin. | Preincubation | 01-138 | |||||
| PKCθ (PRKCQ) | STK | Km bin. | 01-140 | ||||||
| PKCι (PRKCI) | STK | Km bin. | 01-139 | ||||||
| PKD1 (PRKD1) | STK | Km bin. | Preincubation | 02-157 | |||||
| PKD2 (PRKD2) | STK | Km bin. | 1 mM | Preincubation | STK | 02-158 | |||
| PKD3 (PRKD3) | STK | Km bin. | 02-159 | ||||||
| PKN1 | STK | Km bin. | 01-144 | ||||||
| PKR (EIF2AK2) | STK | Km bin. | 05-156 | ||||||
| PLK1 | STK | Km bin. | 1 mM | Cell Cycle | 05-157 | ||||
| PLK2 | STK | Km bin. | Cell Cycle | 05-158 | |||||
| PLK3 | STK | Km bin. | 1 mM | 05-159 | |||||
| PRKX | STK | Km bin. | 01-130 | ||||||
| PYK2 (PTK2B) | TK | Km bin. | 1 mM | Preincubation | TK | 08-138 | |||
| QIK (SNF1LK2) | STK | Km bin. | 1 mM | Preincubation | 02-129 | ||||
| RAF1 | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-125 | |||||
| RET | TK | Km bin. | 1 mM | Preincubation | 08-159 | ||||
| RET[G691S] | TK | Km bin. | 1 mM | Preincubation | 08-522 | ||||
| RET[Y791F] | TK | Km bin. | 1 mM | Preincubation | 08-521 | ||||
| RET[S891A] | TK | Km bin. | 1 mM | Preincubation | 08-523 | ||||
| RET[M918T] | TK | Km bin. | 1 mM | Preincubation | 08-508 | ||||
| ROCK1 | STK | Km bin. | 1 mM | STK | 01-109 | ||||
| ROCK2 | STK | Km bin. | Preincubation | 01-110 | |||||
| RON (MST1R) | TK | Km bin. | 1 mM | Preincubation | 08-152 | ||||
| ROS (ROS1) | TK | Km bin. | 1 mM | Preincubation | 08-163 | ||||
| RSK1(RPS6KA1) | STK | Km bin. | 1 mM | Cell Cycle | 01-149 | ||||
| RSK2 (RPS6KA3) | STK | Km bin. | Preincubation | 01-150 | |||||
| RSK3 (RPS6KA2) | STK | Km bin. | 1 mM | Preincubation | 01-151 | ||||
| RSK4 (RPS6KA6) | STK | Km bin. | 1 mM | Preincubation | 01-152 | ||||
| SGK | STK | Km bin. | 1 mM | Preincubation | STK | 01-158 | |||
| SGK2 | STK | Km bin. | 01-159 | ||||||
| SGK3 (SGKL) | STK | Km bin. | Preincubation | 01-160 | |||||
| SIK (SNF1LK) | STK | Km bin. | 1 mM | 02-131 | |||||
| skMLCK (MYLK2) | STK | Km bin. | 1 mM | Preincubation | 02-150 | ||||
| SLK | STK | Km bin. | 07-129 | ||||||
| SRC | TK | Km bin. | 1 mM | Preincubation | TK | 08-173 | |||
| SRM (SRMS) | TK | Km bin. | 1 mM | Preincubation | 08-174 | ||||
| SRPK1 | STK | Km bin. | 04-160 | ||||||
| SRPK2 | STK | Km bin. | 04-161 | ||||||
| SYK | TK | Km bin. | 1 mM | TK | 08-176 | ||||
| TAK1-TAB1 (MAP3K7) | STK | 1 mM (Cascade) | MAPK (Cascade) | 09-019 | |||||
| TAOK2 | STK | Km bin. | 07-133 | ||||||
| TBK1 | STK | Km bin. | Preincubation | 05-115 | |||||
| TEC | TK | Km bin. | 1 mM | Preincubation | 08-182 | ||||
| TIE2 (TEK) | TK | Km bin. | 1 mM | Preincubation | TK | 08-185 | |||
| TNIK | STK | Km bin. | 1 mM | 07-138 | |||||
| TNK1 | TK | Km bin. | 1 mM | 08-104 | |||||
| TRKA (NTRK1) | TK | Km bin. | 1 mM | TK | 08-186 | ||||
| TRKB (NTRK2) | TK | Km bin. | 1 mM | Preincubation | 08-187 | ||||
| TRKC (NTRK3) | TK | Km bin. | 1 mM | Preincubation | 08-197 | ||||
| TSSK1 | STK | Km bin. | 1 mM | Preincubation | STK | 02-364 | |||
| TSSK2 | STK | Km bin. | 02-165 | ||||||
| TSSK3 | STK | Km bin. | 02-166 | ||||||
| TXK | TK | Km bin. | 1 mM | 08-183 | |||||
| TYK2 | TK | Km bin. | 1 mM | 08-147 | |||||
| TYRO3 | TK | Km bin. | 1 mM | Preincubation | TK | 08-109 | |||
| WNK1 | STK | Km bin. | 05-179 | ||||||
| WNK2 | STK | Km bin. | 05-180 | ||||||
| WNK3 | STK | Km bin. | 05-181 | ||||||
| YES (YES1) | TK | Km bin. | 1 mM | Preincubation | 08-175 | ||||
| YES (YES1) [T348I] | TK | Km bin. | 1 mM | Preincubation | 08-533 | ||||
| ZAP70 | TK | Km bin. | 1 mM | 08-177 | |||||